Cart
sales@molnova.com
PROTAC ERRα ligand 1
CAS No. 1264754-13-3
PROTAC ERRα ligand 1( —— )
Catalog No. M23437 CAS No. 1264754-13-3
PROTAC ERRα ligand 1 is an α (ERRα) antagonist of estrogen-related receptor (IC50s of 0.04 and 2.8 μM for ERRα and ERRγ, respectively).
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 57 | In Stock |
|
| 5MG | 87 | In Stock |
|
| 10MG | 132 | In Stock |
|
| 25MG | 237 | In Stock |
|
| 50MG | 385 | In Stock |
|
| 100MG | 575 | In Stock |
|
| 500MG | 1233 | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
-
Product NamePROTAC ERRα ligand 1
-
NoteResearch use only, not for human use.
-
Brief DescriptionPROTAC ERRα ligand 1 is an α (ERRα) antagonist of estrogen-related receptor (IC50s of 0.04 and 2.8 μM for ERRα and ERRγ, respectively).
-
DescriptionPROTAC ERRα ligand 1 is an α (ERRα) antagonist of estrogen-related receptor (IC50s of 0.04 and 2.8 μM for ERRα and ERRγ, respectively).
-
In Vitro——
-
In Vivo——
-
Synonyms——
-
PathwayEndocrinology/Hormones
-
TargetEstrogen Receptor/ERR
-
RecptorERRα|ERRγ
-
Research Area——
-
Indication——
Chemical Information
-
CAS Number1264754-13-3
-
Formula Weight420.36
-
Molecular FormulaC19H11F3N2O4S
-
Purity>98% (HPLC)
-
SolubilityDMSO : 120 mg/mL (285.47 mM; Need ultrasonic)
-
SMILESN#CC1=CC=C(OC2=CC=C(/C=C(SC(N3)=O)/C3=O)C=C2OC)C(C(F)(F)F)=C1
-
Chemical Name——
Shipping & Storage Information
-
Storage(-20℃)
-
ShippingWith Ice Pack
-
Stability≥ 2 years
Reference
1.Patch RJ, et al. Identification of diaryl ether-based ligands for estrogen-related receptor α as potential antidiabetic agents. J Med Chem. 2011 Feb 10;54(3):788-808.
molnova catalog
related products
-
Diarylpropionitrile
Diarylpropionitrile (DPN) is a non-steroidal estrogen receptor β(ERβ) selective ligand.
-
LSZ102
LSZ102 is a potent, orally bioavailable, selective estrogen receptor degrader (SERD) with ERα transcription IC50 of 6 nM and ERα degradation IC50 of 0.2 nM.
-
Diptoindonesin G
A natural compound, novel chemical probe reciprocally stabilizes ERβ and destabilizes ERα in breast cancer cells.
